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2020
Kroeger, Lukas, Daniliuc, Constantin G. ORCID: 0000-0002-6709-3673, Ensan, Deeba, Borgert, Sebastian, Nienberg, Christian, Lauwers, Miriam, Steinkrueger, Michaela, Jose, Joachim, Pietsch, Markus and Wuensch, Bernhard
(2020).
Synthesis and SAR of Tetracyclic Inhibitors of Protein Kinase CK2 Derived from Furocarbazole W16.
ChemMedChem, 15 (10).
S. 871 - 882.
WEINHEIM:
WILEY-V C H VERLAG GMBH.
ISSN 1860-7187
Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Nickelsen, Anna, Applegate, Violetta M., Jose, Joachim and Niefind, Karsten
ORCID: 0000-0002-0183-6315
(2020).
Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2.
J. Med. Chem., 63 (14).
S. 7766 - 7773.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
Pietsch, Markus, Viht, Kaido, Schnitzler, Alexander, Ekambaram, Ramesh, Steinkrueger, Michaela, Enkvist, Erki, Nienberg, Christian, Nickelsen, Anna, Lauwers, Miriam, Jose, Joachim, Uri, Asko and Niefind, Karsten ORCID: 0000-0002-0183-6315
(2020).
Unexpected CK2 beta-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2.
Bioorganic Chem., 96.
SAN DIEGO:
ACADEMIC PRESS INC ELSEVIER SCIENCE.
ISSN 1090-2120
2019
Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Nickelsen, Anna, Applegate, Violetta M., Hochscherf, Jennifer, Witulski, Benedict, Bouaziz, Zouhair, Marminon, Christelle
ORCID: 0000-0002-4043-3949, Bretner, Maria, Le Borgne, Marc
ORCID: 0000-0003-1398-075X, Jose, Joachim and Niefind, Karsten
ORCID: 0000-0002-0183-6315
(2019).
Diacritic Binding of an Indenoindole Inhibitor by CK2 alpha Paralogs Explored by a Reliable Path to Atomic Resolution CK2 alpha ' Structures.
ACS Omega, 4 (3).
S. 5471 - 5479.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 2470-1343
2018
Schnitzler, Alexander, Gratz, Andreas, Bollacke, Andre, Weyrich, Michael, Kucklaender, Uwe, Wuensch, Bernhard, Goetz, Claudia, Niefind, Karsten ORCID: 0000-0002-0183-6315 and Jose, Joachim
(2018).
A pi-Halogen Bond of Dibenzofuranones with the Gatekeeper Phe113 in Human Protein Kinase CK2 Leads to Potent Tight Binding Inhibitors.
Pharmaceuticals, 11 (1).
BASEL:
MDPI.
ISSN 1424-8247
2017
Hochscherf, Jennifer ORCID: 0000-0002-4412-7391, Lindenblatt, Dirk, Witulski, Benedict, Birus, Robin, Aichele, Dagmar, Marminon, Christelle
ORCID: 0000-0002-4043-3949, Bouaziz, Zouhair, Le Borgne, Marc
ORCID: 0000-0003-1398-075X, Jose, Joachim and Niefind, Karsten
ORCID: 0000-0002-0183-6315
(2017).
Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2 alpha and Its Paralog CK2 alpha '.
Pharmaceuticals, 10 (4).
BASEL:
MDPI.
ISSN 1424-8247