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2020
Wodtke, Robert, Pietsch, Markus and Loeser, Reik (2020). Solution-phase synthesis of the fluorogenic TGase 2 acyl donor Z-Glu(HMC)-Gly-OH and its use for inhibitor and amine substrate characterisation. Anal. Biochem., 595. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1096-0309
2018
Wodtke, Robert ORCID: 0000-0001-7462-7111, Hauser, Christoph, Ruiz-Gomez, Gloria, Jaeckel, Elisabeth, Bauer, David, Lohse, Martin, Wong, Alan, Pufe, Johanna, Ludwig, Friedrich-Alexander, Fischer, Steffen, Hauser, Sandra
ORCID: 0000-0001-8206-6000, Greif, Dieter, Pisabarro, M. Teresa, Pietzsch, Jens
ORCID: 0000-0002-1610-1493, Pietsch, Markus and Loeser, Reik
(2018).
N-epsilon-Acryloyllysine Piperazides as Irreversible Inhibitors of Transglutaminase 2: Synthesis, Structure-Activity Relationships, and Pharmacokinetic Profiling.
J. Med. Chem., 61 (10).
S. 4528 - 4561.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
2017
Hauser, Christoph, Wodtke, Robert ORCID: 0000-0001-7462-7111, Loeser, Reik and Pietsch, Markus
(2017).
A fluorescence anisotropy-based assay for determining the activity of tissue transglutaminase.
Amino Acids, 49 (3).
S. 567 - 584.
WIEN:
SPRINGER WIEN.
ISSN 1438-2199
2016
Wodtke, Robert ORCID: 0000-0001-7462-7111, Schramm, Georg
ORCID: 0000-0002-2251-3195, Pietzsch, Jens
ORCID: 0000-0002-1610-1493, Pietsch, Markus and Loeser, Reik
(2016).
Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminase 2.
ChemBioChem, 17 (13).
S. 1263 - 1282.
WEINHEIM:
WILEY-V C H VERLAG GMBH.
ISSN 1439-7633
2015
Hauser, Christoph, Wodtke, Robert, Loeser, Reik and Pietsch, Markus (2015). A new fluorescence anisotropy-based assay for activity determination of tissue transglutaminase. Amino Acids, 47 (8). S. 1629 - 1630. WIEN: SPRINGER WIEN. ISSN 1438-2199