![]() | Up a level |
Journal Article
Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Applegate, Violetta
ORCID: 0000-0003-4120-7983, Nickelsen, Anna, Klussmann, Merlin, Neundorf, Ines, Goetz, Claudia, Jose, Joachim
ORCID: 0000-0002-0666-2676 and Niefind, Karsten
ORCID: 0000-0002-0183-6315
(2022).
Molecular Plasticity of Crystalline CK2 alpha ' Leads to KN2, a Bivalent Inhibitor of Protein Kinase CK2 with Extraordinary Selectivity.
J. Med. Chem., 65 (2).
S. 1302 - 1313.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Nickelsen, Anna, Applegate, Violetta M., Jose, Joachim and Niefind, Karsten
ORCID: 0000-0002-0183-6315
(2020).
Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2.
J. Med. Chem., 63 (14).
S. 7766 - 7773.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Horn, Mareike, Goetz, Claudia, Niefind, Karsten
ORCID: 0000-0002-0183-6315, Neundorf, Ines
ORCID: 0000-0001-6450-3991 and Pietsch, Markus
(2019).
Design of CK2 beta-Mimicking Peptides as Tools To Study the CK2 alpha/CK2 beta Interaction in Cancer Cells.
ChemMedChem, 14 (8).
S. 833 - 842.
WEINHEIM:
WILEY-V C H VERLAG GMBH.
ISSN 1860-7187
Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Nickelsen, Anna, Applegate, Violetta M., Hochscherf, Jennifer, Witulski, Benedict, Bouaziz, Zouhair, Marminon, Christelle
ORCID: 0000-0002-4043-3949, Bretner, Maria, Le Borgne, Marc
ORCID: 0000-0003-1398-075X, Jose, Joachim and Niefind, Karsten
ORCID: 0000-0002-0183-6315
(2019).
Diacritic Binding of an Indenoindole Inhibitor by CK2 alpha Paralogs Explored by a Reliable Path to Atomic Resolution CK2 alpha ' Structures.
ACS Omega, 4 (3).
S. 5471 - 5479.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 2470-1343
Thesis
Lindenblatt, Dirk ORCID: 0000-0002-5561-1082
(2022).
Structural Exploration of Different Binding Pockets Suitable to Affect Protein Kinases CK2α and CK2α’ With Peptides and Small Molecules.
PhD thesis, Universität zu Köln.