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Number of items: 9.

Journal Article

Asif, Maria, Kaygusuz, Emrah, Shinawi, Marwan, Nickelsen, Anna, Hsieh, Tzung-Chien, Wagle, Prerana, Budde, Birgit S., Hochscherf, Jennifer ORCID: 0000-0002-4412-7391, Abdullah, Uzma, Honing, Stefan, Nienberg, Christian, Lindenblatt, Dirk, Noegel, Angelika A., Altmuller, Janine ORCID: 0000-0003-4372-1521, Thiele, Holger, Motameny, Susanne, Fleischer, Nicole, Segal, Idan, Pais, Lynn, Tinschert, Sigrid, Samra, Nadra Nasser, Savatt, Juliann M., Rudy, Natasha L., De Luca, Chiara, Fortugno, Paola, White, Susan M., Krawitz, Peter, Hurst, Anna C. E., Niefind, Karsten ORCID: 0000-0002-0183-6315, Jose, Joachim ORCID: 0000-0002-0666-2676, Brancati, Francesco, Nurnberg, Peter and Hussain, Muhammad Sajid ORCID: 0000-0002-1353-8809 (2022). De novo variants of CSNK2B cause a new intellectual disability-craniodigital syndrome by disrupting the canonical Wnt signaling pathway. Hum. Genet. Genom. Adv., 3 (3). AMSTERDAM: ELSEVIER. ISSN 2666-2477

Hochscherf, Jennifer ORCID: 0000-0002-4412-7391, Lindenblatt, Dirk, Witulski, Benedict, Birus, Robin, Aichele, Dagmar, Marminon, Christelle ORCID: 0000-0002-4043-3949, Bouaziz, Zouhair, Le Borgne, Marc ORCID: 0000-0003-1398-075X, Jose, Joachim and Niefind, Karsten ORCID: 0000-0002-0183-6315 (2017). Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2 alpha and Its Paralog CK2 alpha '. Pharmaceuticals, 10 (4). BASEL: MDPI. ISSN 1424-8247

Kroeger, Lukas, Daniliuc, Constantin G. ORCID: 0000-0002-6709-3673, Ensan, Deeba, Borgert, Sebastian, Nienberg, Christian, Lauwers, Miriam, Steinkrueger, Michaela, Jose, Joachim, Pietsch, Markus and Wuensch, Bernhard (2020). Synthesis and SAR of Tetracyclic Inhibitors of Protein Kinase CK2 Derived from Furocarbazole W16. ChemMedChem, 15 (10). S. 871 - 882. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1860-7187

Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Applegate, Violetta ORCID: 0000-0003-4120-7983, Nickelsen, Anna, Klussmann, Merlin, Neundorf, Ines, Goetz, Claudia, Jose, Joachim ORCID: 0000-0002-0666-2676 and Niefind, Karsten ORCID: 0000-0002-0183-6315 (2022). Molecular Plasticity of Crystalline CK2 alpha ' Leads to KN2, a Bivalent Inhibitor of Protein Kinase CK2 with Extraordinary Selectivity. J. Med. Chem., 65 (2). S. 1302 - 1313. WASHINGTON: AMER CHEMICAL SOC. ISSN 1520-4804

Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Nickelsen, Anna, Applegate, Violetta M., Hochscherf, Jennifer, Witulski, Benedict, Bouaziz, Zouhair, Marminon, Christelle ORCID: 0000-0002-4043-3949, Bretner, Maria, Le Borgne, Marc ORCID: 0000-0003-1398-075X, Jose, Joachim and Niefind, Karsten ORCID: 0000-0002-0183-6315 (2019). Diacritic Binding of an Indenoindole Inhibitor by CK2 alpha Paralogs Explored by a Reliable Path to Atomic Resolution CK2 alpha ' Structures. ACS Omega, 4 (3). S. 5471 - 5479. WASHINGTON: AMER CHEMICAL SOC. ISSN 2470-1343

Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Nickelsen, Anna, Applegate, Violetta M., Jose, Joachim and Niefind, Karsten ORCID: 0000-0002-0183-6315 (2020). Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2. J. Med. Chem., 63 (14). S. 7766 - 7773. WASHINGTON: AMER CHEMICAL SOC. ISSN 1520-4804

Pietsch, Markus, Viht, Kaido, Schnitzler, Alexander, Ekambaram, Ramesh, Steinkrueger, Michaela, Enkvist, Erki, Nienberg, Christian, Nickelsen, Anna, Lauwers, Miriam, Jose, Joachim, Uri, Asko and Niefind, Karsten ORCID: 0000-0002-0183-6315 (2020). Unexpected CK2 beta-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2. Bioorganic Chem., 96. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1090-2120

Schnitzler, Alexander, Gratz, Andreas, Bollacke, Andre, Weyrich, Michael, Kucklaender, Uwe, Wuensch, Bernhard, Goetz, Claudia, Niefind, Karsten ORCID: 0000-0002-0183-6315 and Jose, Joachim (2018). A pi-Halogen Bond of Dibenzofuranones with the Gatekeeper Phe113 in Human Protein Kinase CK2 Leads to Potent Tight Binding Inhibitors. Pharmaceuticals, 11 (1). BASEL: MDPI. ISSN 1424-8247

Werner, Christian, Gast, Alexander, Lindenblatt, Dirk, Nickelsen, Anna, Niefind, Karsten ORCID: 0000-0002-0183-6315, Jose, Joachim ORCID: 0000-0002-0666-2676 and Hochscherf, Jennifer ORCID: 0000-0002-4412-7391 (2022). Structural and Enzymological Evidence for an Altered Substrate Specificity in Okur-Chung Neurodevelopmental Syndrome Mutant CK2 alpha(Lys198Arg). Front. Mol. Biosci., 9. LAUSANNE: FRONTIERS MEDIA SA. ISSN 2296-889X

This list was generated on Fri Mar 29 05:53:39 2024 CET.