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Braegelmann, Johannes, Dammert, Marcel A., Dietlein, Felix, Heuckmann, Johannes M., Choidas, Axel, Boehm, Stefanie, Richters, Andre, Basu, Debjit, Tischler, Verena ORCID: 0000-0002-6673-8329, Lorenz, Carina, Habenberger, Peter, Fang, Zhizhou, Ortiz-Cuaran, Sandra, Leenders, Frauke, Eickhoff, Jan, Koch, Uwe, Getlik, Matthaeus, Termathe, Martin
ORCID: 0000-0002-5618-4633, Sallouh, Muhammad, Greff, Zoltan, Varga, Zoltan, Balke-Want, Hyatt, French, Christopher A., Peifer, Martin
ORCID: 0000-0002-5243-5503, Reinhardt, H. Christian, Orfi, Laszlo
ORCID: 0000-0001-6149-2385, Keri, Gyorgy, Ansen, Sascha, Heukamp, Lukas C., Buettner, Reinhard, Rauh, Daniel, Klebl, Bert M., Thomas, Roman K. and Sos, Martin L.
(2017).
Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma.
Cell Reports, 20 (12).
S. 2833 - 2846.
CAMBRIDGE:
CELL PRESS.
ISSN 2211-1247
Dietlein, Felix, Kalb, Bastian, Jokic, Mladen, Noll, Elisa M., Strong, Alexander, Tharun, Lars, Ozretic, Luka, Kuenstlinger, Helen, Kambartel, Kato, Randerath, Winfried J., Juengst, Christian, Schmitt, Anna, Torgovnick, Alessandro, Richters, Andre, Rauh, Daniel ORCID: 0000-0002-1970-7642, Siedek, Florian, Persigehl, Thorsten, Mauch, Cornelia, Bartkova, Jirina, Bradley, Allan
ORCID: 0000-0002-2349-8839, Sprick, Martin R.
ORCID: 0000-0001-9691-7574, Trumpp, Andreas
ORCID: 0000-0002-6212-3466, Rad, Roland, Saur, Dieter
ORCID: 0000-0001-5874-0210, Bartek, Jiri, Wolf, Juergen, Buettner, Reinhard, Thomas, Roman K. and Reinhardt, H. Christian
(2015).
A Synergistic Interaction between Chk1-and MK2 Inhibitors in KRAS-Mutant Cancer.
Cell, 162 (1).
S. 146 - 160.
CAMBRIDGE:
CELL PRESS.
ISSN 1097-4172
Engel, Julian, Richters, Andre, Getlik, Matthaeus, Tomassi, Stefano, Keul, Marina, Termathe, Martin ORCID: 0000-0002-5618-4633, Lategahn, Jonas
ORCID: 0000-0001-5993-7082, Becker, Christian, Mayer-Wrangowski, Svenja, Gruetter, Christian, Uhlenbrock, Niklas
ORCID: 0000-0002-4489-9535, Kruell, Jasmin, Schaumann, Niklas, Eppmann, Simone, Kibies, Patrick, Hoffgaard, Franziska, Heil, Jochen, Menninger, Sascha, Ortiz-Cuaran, Sandra, Heuckmann, Johannes M., Tinnefeld, Verena, Zahedi, Rene P., Sos, Martin L., Schultz-Fademrecht, Carsten, Thomas, Roman K., Kast, Stefan M. and Rauh, Daniel
ORCID: 0000-0002-1970-7642
(2015).
Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach.
J. Med. Chem., 58 (17).
S. 6844 - 6864.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
Malchers, Florian, Dietlein, Felix, Schottle, Jakob, Lu, Xin, Nogova, Lucia, Albus, Kerstin, Fernandez-Cuesta, Lynnette ORCID: 0000-0002-0724-6703, Heuckmann, Johannes M., Gautschi, Oliver, Diebold, Joachim, Plenker, Dennis, Gardizi, Masyar, Er, Matthias Scheffl, Bos, Marc, Seidel, Danila, Leenders, Frauke, Richters, Andre, Peifer, Martin
ORCID: 0000-0002-5243-5503, Florin, Alexandra, Mainkar, Prathama S., Karre, Nagaraju, Chandrasekhar, Srivari, George, Julie, Silling, Steffi, Rauh, Daniel
ORCID: 0000-0002-1970-7642, Zander, Thomas, Ullrich, Roland T., Reinhardt, H. Christian, Ringeisen, Francois, Buettner, Reinhard, Heukamp, Lukas C., Wolf, Juergen and Thomas, Roman K.
(2014).
Cell-Autonomous and Non-Cell-Autonomous Mechanisms of Transformation by Amplified FGFR1 in Lung Cancer.
Cancer Discov., 4 (2).
S. 246 - 258.
PHILADELPHIA:
AMER ASSOC CANCER RESEARCH.
ISSN 2159-8290
Plenker, Dennis, Riedel, Maximilian, Braegelmann, Johannes, Dammert, Marcel A., Chauhan, Rakhee, Knowles, Phillip P., Lorenz, Carina, Keul, Marina, Buehrmann, Mike, Pagel, Oliver, Tischler, Verena ORCID: 0000-0002-6673-8329, Scheel, Andreas H., Schtte, Daniel, Song, Yanrui, Stark, Justina, Mrugalla, Florian
ORCID: 0000-0002-6281-6051, Alber, Yannic, Richters, Andre, Engel, Julian, Leenders, Frauke, Heuckmann, Johannes M., Wolf, Juergen, Diebold, Joachim, Pall, Georg, Peifer, Martin
ORCID: 0000-0002-5243-5503, Aerts, Maarten, Gevaert, Kris
ORCID: 0000-0002-4237-0283, Zahedi, Rene P., Buettner, Reinhard, Shokat, Kevan M., McDonald, Neil Q., Kast, Stefan M., Gautschi, Oliver, Thomas, Roman K. and Sos, Martin L.
(2017).
Drugging the catalytically inactive state of RET kinase in RET-rearranged tumors.
Sci. Transl. Med., 9 (394).
WASHINGTON:
AMER ASSOC ADVANCEMENT SCIENCE.
ISSN 1946-6242
Richters, Andre, Basu, Debjit, Engel, Julian, Ercanoglu, Meryem S., Balke-Want, Hyatt, Tesch, Roberta, Thomas, Roman K. and Rauh, Daniel ORCID: 0000-0002-1970-7642
(2015).
Identification and Further Development of Potent TBK1 Inhibitors.
ACS Chem. Biol., 10 (1).
S. 289 - 299.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1554-8937
Sos, Martin L., Dietlein, Felix, Peifer, Martin ORCID: 0000-0002-5243-5503, Schoettle, Jakob, Balke-Want, Hyatt, Mueller, Christian, Koker, Mirjam, Richters, Andre, Heynck, Stefanie, Malchers, Florian, Heuckmann, Johannes M., Seidel, Danila, Eyers, Patrick A., Ullrich, Roland T., Antonchick, Andrey P., Vintonyak, Viktor V., Schneider, Peter M.
ORCID: 0000-0003-0744-2349, Ninomiya, Takashi, Waldmann, Herbert
ORCID: 0000-0002-9606-7247, Buettner, Reinhard, Rauh, Daniel
ORCID: 0000-0002-1970-7642, Heukamp, Lukas C. and Thomas, Roman K.
(2012).
A framework for identification of actionable cancer genome dependencies in small cell lung cancer.
Proc. Natl. Acad. Sci. U. S. A., 109 (42).
S. 17034 - 17040.
WASHINGTON:
NATL ACAD SCIENCES.
ISSN 0027-8424