Universität zu Köln

Akhtar-Schaefer, Isha, Reuten, Raphael, Koch, Manuel, Pietsch, Markus and Langmann, Thomas (2019). AMD-Associated HTRA1 Variants Do Not Influence TGF-beta Signaling in Microglia. S. 3 - 8. CHAM: SPRINGER INTERNATIONAL PUBLISHING AG. ISSN 2214-8019

Baeuml, Charlotte A., George, Ajay Abisheck Paul, Schmitz, Thomas, Sommerfeld, Paul, Pietsch, Markus, Podsiadlowski, Lars, Steinmetzer, Torsten, Biswas, Arijit and Imhof, Diana (2020). Distinct 3-disulfide-bonded isomers of tridegin differentially inhibit coagulation factor XIIIa: The influence of structural stability on bioactivity. Eur. J. Med. Chem., 201. ISSY-LES-MOULINEAUX: ELSEVIER FRANCE-EDITIONS SCIENTIFIQUES MEDICALES ELSEVIER. ISSN 1768-3254

Braeutigam, Maria, Teusch, Nicole ORCID: 0000-0002-9030-1493, Schenk, Tobias, Sheikh, Miriam, Aricioglu, Rocky Z., Borowski, Swantje H., Neudoerfl, Joerg-Martin, Baumann, Ulrich, Griesbeck, Axel G. and Pietsch, Markus (2015). Selective Inhibitors of Glutathione Transferase P1 with Trioxane Structure as Anticancer Agents. ChemMedChem, 10 (4). S. 629 - 640. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1860-7187

Braeutigam, Maria, Teusch, Nicole ORCID: 0000-0002-9030-1493, Schenk, Tobias, Sheikh, Miriam, Aricioglu, Rocky Z., Borowski, Swantje H., Neudoerfl, Joerg-Martin, Baumann, Ulrich, Griesbeck, Axel G. and Pietsch, Markus (2015). Selective Inhibitors of Glutathione Transferase P1 with Trioxane Structure as Anticancer Agents. ChemMedChem, 10 (4). S. 629 - 640. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1860-7187

Dahlinger, Dominik, Aslan, Sevinc, Pietsch, Markus, Frechen, Sebastian and Fuhr, Uwe (2017). Assessment of inhibitory effects on major human cytochrome P450 enzymes by spasmolytics used in the treatment of overactive bladder syndrome. Ther. Adv. Urol., 9 (7). S. 163 - 178. LONDON: SAGE PUBLICATIONS LTD. ISSN 1756-2880

Dato, Florian M., Maassen, Andreas ORCID: 0000-0002-1446-0994, Goldfuss, Bernd ORCID: 0000-0002-1814-8818 and Pietsch, Markus (2018). Characterization of fatty acid amide hydrolase activity by a fluorescence-based assay. Anal. Biochem., 546. S. 50 - 58. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1096-0309

Dato, Florian M., Neudoerfl, Jorg-Martin, Guetschow, Michael, Goldfuss, Bernd ORCID: 0000-0002-1814-8818 and Pietsch, Markus (2020). omega-Quinazolinonylalkyl aryl ureas as reversible inhibitors of monoacylglycerol lipase. Bioorganic Chem., 94. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1090-2120

Dato, Florian M., Sheikh, Miriam, Uhl, Rocky Z., Schueller, Alexandra W., Steinkrueger, Michaela, Koch, Peter, Neudoerfl, Joerg-Martin, Guetschow, Michael, Goldfuss, Bernd ORCID: 0000-0002-1814-8818 and Pietsch, Markus (2018). omega -Phthalimidoalkyl Aryl Ureas as Potent and Selective Inhibitors of Cholesterol Esterase. ChemMedChem, 13 (17). S. 1833 - 1848. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1860-7187

El-Awaad, Ehab, Pryymachuk, Galyna, Fried, Cora, Matthes, Jan ORCID: 0000-0003-2754-1555, Isensee, Joerg, Hucho, Tim, Neiss, Wolfram F., Paulsson, Mats, Herzig, Stefan, Zaucke, Frank and Pietsch, Markus (2019). Direct, gabapentin-insensitive interaction of a soluble form of the calcium channel subunit alpha(2)delta-1 with thrombospondin-4. Sci Rep, 9. LONDON: NATURE PUBLISHING GROUP. ISSN 2045-2322

Griesbeck, Axel G. ORCID: 0000-0002-6546-3482, Maassen, Andreas ORCID: 0000-0002-1446-0994, Braeutigam, Maria and Pietsch, Markus (2015). Model Studies on Peroxidic Glutathione Transferase (GST) Inhibitors: C5-Methylated 1,2,4-Trioxanes with C6-Acrylate Side Chains. Eur. J. Org. Chem., 2015 (20). S. 4349 - 4353. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1099-0690

Hauser, Christoph, Wodtke, Robert ORCID: 0000-0001-7462-7111, Loeser, Reik and Pietsch, Markus (2017). A fluorescence anisotropy-based assay for determining the activity of tissue transglutaminase. Amino Acids, 49 (3). S. 567 - 584. WIEN: SPRINGER WIEN. ISSN 1438-2199

Hauser, Christoph, Wodtke, Robert, Loeser, Reik and Pietsch, Markus (2015). A new fluorescence anisotropy-based assay for activity determination of tissue transglutaminase. Amino Acids, 47 (8). S. 1629 - 1630. WIEN: SPRINGER WIEN. ISSN 1438-2199

Hauser, Sandra ORCID: 0000-0001-8206-6000, Sommerfeld, Paul ORCID: 0000-0002-8182-0347, Wodtke, Johanna, Hauser, Christoph ORCID: 0000-0003-4103-5843, Schlitterlau, Paul, Pietzsch, Jens ORCID: 0000-0002-1610-1493, Loeser, Reik, Pietsch, Markus ORCID: 0000-0002-8110-2265 and Wodtke, Robert ORCID: 0000-0001-7462-7111 (2022). Application of a Fluorescence Anisotropy-Based Assay to Quantify Transglutaminase 2 Activity in Cell Lysates. Int. J. Mol. Sci., 23 (9). BASEL: MDPI. ISSN 1422-0067

Heng, Sabrina, Tieu, William ORCID: 0000-0002-7161-4152, Hautmann, Stephanie, Kuan, Kevin, Pedersen, Daniel Sejer ORCID: 0000-0003-3926-7047, Pietsch, Markus, Guetschow, Michael and Abell, Andrew D. (2011). New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds. Bioorg. Med. Chem., 19 (24). S. 7453 - 7464. OXFORD: PERGAMON-ELSEVIER SCIENCE LTD. ISSN 1464-3391

Hochscherf, Jennifer ORCID: 0000-0002-4412-7391, Lindenblatt, Dirk, Steinkrtiger, Michaela, Yoo, Eungyoung, Ulucan, Oezlem, Herzig, Stefan, Issinger, Olaf-Georg, Helms, Volkhard ORCID: 0000-0002-2180-9154, Goetz, Claudia, Neundorf, Ines ORCID: 0000-0001-6450-3991, Niefind, Karsten ORCID: 0000-0002-0183-6315 and Pietsch, Markus (2015). Development of a high-throughput screening-compatible assay to identify inhibitors of the CK2 alpha/CK2 beta interaction. Anal. Biochem., 468. S. 4 - 15. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1096-0309

Hochscherf, Jennifer ORCID: 0000-0002-4412-7391, Pietsch, Markus, Tieu, William ORCID: 0000-0002-7161-4152, Kuan, Kevin, Abell, Andrew D., Guetschow, Michael and Niefind, Karsten ORCID: 0000-0002-0183-6315 (2018). Crystal structure of highly glycosylated human leukocyte elastase in complex with an S2 ' site binding inhibitor. Acta Crystallogr. F-Struct. Biol. Commun., 74. S. 480 - 490. CHESTER: INT UNION CRYSTALLOGRAPHY. ISSN 2053-230X

Kroeger, Lukas, Daniliuc, Constantin G. ORCID: 0000-0002-6709-3673, Ensan, Deeba, Borgert, Sebastian, Nienberg, Christian, Lauwers, Miriam, Steinkrueger, Michaela, Jose, Joachim, Pietsch, Markus and Wuensch, Bernhard (2020). Synthesis and SAR of Tetracyclic Inhibitors of Protein Kinase CK2 Derived from Furocarbazole W16. ChemMedChem, 15 (10). S. 871 - 882. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1860-7187

Lemke, Carina, Christmann, Joscha, Yin, Jiafei, Alonso, Jose M., Serrano, Estefania, Chioua, Mourad, Ismaili, Lhassane, Angeles Martinez-Grau, Maria, Beadle, Christopher D., Vetman, Tatiana, Dato, Florian M., Bartz, Ulrike, Elsinghorst, Paul W., Pietsch, Markus, Mueller, Christa E., Iriepa, Isabel ORCID: 0000-0003-3475-9624, Wille, Timo ORCID: 0000-0002-4359-5388, Marco-Contelles, Jose and Guetschow, Michael (2019). Chromenones as Multineurotargeting Inhibitors of Human Enzymes. ACS Omega, 4 (26). S. 22161 - 22169. WASHINGTON: AMER CHEMICAL SOC. ISSN 2470-1343

Lindenblatt, Dirk ORCID: 0000-0002-5561-1082, Horn, Mareike, Goetz, Claudia, Niefind, Karsten ORCID: 0000-0002-0183-6315, Neundorf, Ines ORCID: 0000-0001-6450-3991 and Pietsch, Markus (2019). Design of CK2 beta-Mimicking Peptides as Tools To Study the CK2 alpha/CK2 beta Interaction in Cancer Cells. ChemMedChem, 14 (8). S. 833 - 842. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1860-7187

Pehere, Ashok, Pietsch, Markus, Paul, Neilsen, Callen, David, Gutschow, Michael and Abell, Andrew (2015). Design, synthesis, and testing of macrocyclic beta-strand as protease inhibitors. Abstr. Pap. Am. Chem. Soc., 249. WASHINGTON: AMER CHEMICAL SOC. ISSN 0065-7727

Pehere, Ashok, Pietsch, Markus, Paul, Neilsen, Callen, David, Gutschow, Michael and Abell, Andrew (2015). Design, synthesis, and testing of macrocyclic beta-strand as protease inhibitors. Abstr. Pap. Am. Chem. Soc., 249. WASHINGTON: AMER CHEMICAL SOC. ISSN 0065-7727

Pepanian, Anna, Sommerfeld, Paul ORCID: 0000-0002-8182-0347, Kasprzyk, Renata, Kuehl, Toni, Binbay, F. Ayberk, Hauser, Christoph, Loeser, Reik, Wodtke, Robert, Bednarczyk, Marcelina, Chrominski, Mikolaj, Kowalska, Joanna, Jemielity, Jacek ORCID: 0000-0001-7633-788X, Imhof, Diana and Pietsch, Markus (2022). Fluorescence Anisotropy Assay with Guanine Nucleotides Provides Access to Functional Analysis of G alpha i1 Proteins. Anal. Chem., 94 (41). S. 14410 - 14419. WASHINGTON: AMER CHEMICAL SOC. ISSN 1520-6882

Pietsch, Markus, Viht, Kaido, Schnitzler, Alexander, Ekambaram, Ramesh, Steinkrueger, Michaela, Enkvist, Erki, Nienberg, Christian, Nickelsen, Anna, Lauwers, Miriam, Jose, Joachim, Uri, Asko and Niefind, Karsten ORCID: 0000-0002-0183-6315 (2020). Unexpected CK2 beta-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2. Bioorganic Chem., 96. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1090-2120

Pietsch, Markus, Wodtke, Robert ORCID: 0000-0001-7462-7111, Pietzsch, Jens ORCID: 0000-0002-1610-1493 and Loeser, Reik (2013). Tissue transglutaminase: An emerging target for therapy and imaging. Bioorg. Med. Chem. Lett., 23 (24). S. 6528 - 6544. OXFORD: PERGAMON-ELSEVIER SCIENCE LTD. ISSN 1464-3405

Pryymachuk, Galyna, El-Awaad, Ehab ORCID: 0000-0003-3383-6384, Piekarek, Nadin, Drebber, Uta, Maul, Alexandra C., Hescheler, Juergen, Wodarz, Andreas ORCID: 0000-0002-0007-6289, Pfitzer, Gabriele, Neiss, Wolfram F., Pietsch, Markus ORCID: 0000-0002-8110-2265 and Schroeter, Mechthild M. (2022). Angiotensin II type 1 receptor localizes at the blood-bile barrier in humans and pigs. Histochem. Cell Biol., 157 (5). S. 513 - 525. NEW YORK: SPRINGER. ISSN 1432-119X

Schaekel, Laura, Mirza, Salahuddin, Pietsch, Markus ORCID: 0000-0002-8110-2265, Lee, Sang-Yong, Keuler, Tim, Sylvester, Katharina, Pelletier, Julie, Sevigny, Jean ORCID: 0000-0003-2922-1600, Pillaiyar, Thanigaimalai, Namasivayam, Vigneshwaran ORCID: 0000-0003-3031-3377, Guetschow, Michael and Mueller, Christa E. (2021). 2-Substituted thienotetrahydropyridine derivatives: Allosteric ectonucleotidase inhibitors. Arch. Pharm., 354 (12). WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1521-4184

Schomaecker, Klaus, Marmann, Verena, Pietsch, Markus, Kirsch, Stefan, Jaschinski, Marcel, Fischer, Thomas and Drzezga, Alexander (2020). Structure-affinity relationships of estrogen derivatives to ER alpha as precursors for radiolabeling in endoradiotherapy of ER-positive mammary carcinomas. J. Nucl. Med., 61. RESTON: SOC NUCLEAR MEDICINE INC. ISSN 1535-5667

Wodtke, Robert ORCID: 0000-0001-7462-7111, Hauser, Christoph, Ruiz-Gomez, Gloria, Jaeckel, Elisabeth, Bauer, David, Lohse, Martin, Wong, Alan, Pufe, Johanna, Ludwig, Friedrich-Alexander, Fischer, Steffen, Hauser, Sandra ORCID: 0000-0001-8206-6000, Greif, Dieter, Pisabarro, M. Teresa, Pietzsch, Jens ORCID: 0000-0002-1610-1493, Pietsch, Markus and Loeser, Reik (2018). N-epsilon-Acryloyllysine Piperazides as Irreversible Inhibitors of Transglutaminase 2: Synthesis, Structure-Activity Relationships, and Pharmacokinetic Profiling. J. Med. Chem., 61 (10). S. 4528 - 4561. WASHINGTON: AMER CHEMICAL SOC. ISSN 1520-4804

Wodtke, Robert, Pietsch, Markus and Loeser, Reik (2020). Solution-phase synthesis of the fluorogenic TGase 2 acyl donor Z-Glu(HMC)-Gly-OH and its use for inhibitor and amine substrate characterisation. Anal. Biochem., 595. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1096-0309

Wodtke, Robert ORCID: 0000-0001-7462-7111, Schramm, Georg ORCID: 0000-0002-2251-3195, Pietzsch, Jens ORCID: 0000-0002-1610-1493, Pietsch, Markus and Loeser, Reik (2016). Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminase 2. ChemBioChem, 17 (13). S. 1263 - 1282. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1439-7633

Wodtke, Robert, Wodtke, Johanna, Hauser, Sandra ORCID: 0000-0001-8206-6000, Laube, Markus, Bauer, David, Rothe, Rebecca ORCID: 0000-0002-0615-1112, Neuber, Christin, Pietsch, Markus, Kopka, Klaus, Pietzsch, Jens ORCID: 0000-0002-1610-1493 and Loeser, Reik (2021). Development of an F-18-Labeled Irreversible Inhibitor of Transglutaminase 2 as Radiometric Tool for Quantitative Expression Profiling in Cells and Tissues. J. Med. Chem., 64 (6). S. 3462 - 3479. WASHINGTON: AMER CHEMICAL SOC. ISSN 1520-4804