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Becker, Christian, Oecal, Sinan, Nguyen, Hoang D., Keul, Marina, Simard, Jeffrey R. and Rauh, Daniel ORCID: 0000-0002-1970-7642
(2016).
Monitoring Conformational Changes in the Receptor Tyrosine Kinase EGFR.
ChemBioChem, 17 (11).
S. 990 - 995.
WEINHEIM:
WILEY-V C H VERLAG GMBH.
ISSN 1439-7633
Braegelmann, Johannes, Dammert, Marcel A., Dietlein, Felix, Heuckmann, Johannes M., Choidas, Axel, Boehm, Stefanie, Richters, Andre, Basu, Debjit, Tischler, Verena ORCID: 0000-0002-6673-8329, Lorenz, Carina, Habenberger, Peter, Fang, Zhizhou, Ortiz-Cuaran, Sandra, Leenders, Frauke, Eickhoff, Jan, Koch, Uwe, Getlik, Matthaeus, Termathe, Martin
ORCID: 0000-0002-5618-4633, Sallouh, Muhammad, Greff, Zoltan, Varga, Zoltan, Balke-Want, Hyatt, French, Christopher A., Peifer, Martin
ORCID: 0000-0002-5243-5503, Reinhardt, H. Christian, Orfi, Laszlo
ORCID: 0000-0001-6149-2385, Keri, Gyorgy, Ansen, Sascha, Heukamp, Lukas C., Buettner, Reinhard, Rauh, Daniel, Klebl, Bert M., Thomas, Roman K. and Sos, Martin L.
(2017).
Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma.
Cell Reports, 20 (12).
S. 2833 - 2846.
CAMBRIDGE:
CELL PRESS.
ISSN 2211-1247
Dietlein, Felix, Kalb, Bastian, Jokic, Mladen, Noll, Elisa M., Strong, Alexander, Tharun, Lars, Ozretic, Luka, Kuenstlinger, Helen, Kambartel, Kato, Randerath, Winfried J., Juengst, Christian, Schmitt, Anna, Torgovnick, Alessandro, Richters, Andre, Rauh, Daniel ORCID: 0000-0002-1970-7642, Siedek, Florian, Persigehl, Thorsten, Mauch, Cornelia, Bartkova, Jirina, Bradley, Allan
ORCID: 0000-0002-2349-8839, Sprick, Martin R.
ORCID: 0000-0001-9691-7574, Trumpp, Andreas
ORCID: 0000-0002-6212-3466, Rad, Roland, Saur, Dieter
ORCID: 0000-0001-5874-0210, Bartek, Jiri, Wolf, Juergen, Buettner, Reinhard, Thomas, Roman K. and Reinhardt, H. Christian
(2015).
A Synergistic Interaction between Chk1-and MK2 Inhibitors in KRAS-Mutant Cancer.
Cell, 162 (1).
S. 146 - 160.
CAMBRIDGE:
CELL PRESS.
ISSN 1097-4172
Engel, Julian, Richters, Andre, Getlik, Matthaeus, Tomassi, Stefano, Keul, Marina, Termathe, Martin ORCID: 0000-0002-5618-4633, Lategahn, Jonas
ORCID: 0000-0001-5993-7082, Becker, Christian, Mayer-Wrangowski, Svenja, Gruetter, Christian, Uhlenbrock, Niklas
ORCID: 0000-0002-4489-9535, Kruell, Jasmin, Schaumann, Niklas, Eppmann, Simone, Kibies, Patrick, Hoffgaard, Franziska, Heil, Jochen, Menninger, Sascha, Ortiz-Cuaran, Sandra, Heuckmann, Johannes M., Tinnefeld, Verena, Zahedi, Rene P., Sos, Martin L., Schultz-Fademrecht, Carsten, Thomas, Roman K., Kast, Stefan M. and Rauh, Daniel
ORCID: 0000-0002-1970-7642
(2015).
Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach.
J. Med. Chem., 58 (17).
S. 6844 - 6864.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
Engel, Julian, Smith, Steven, Lategahn, Jonas ORCID: 0000-0001-5993-7082, Turnbrink, Hannah L., Goebel, Lisa, Becker, Christian, Hennes, Elisabeth, Keul, Marina, Unger, Anke, Mueller, Heiko, Baumann, Matthias, Schultz-Fademrecht, Carsten, Guenther, Georgia, Hengstler, Jan G. and Rauh, Daniel
(2017).
Structure-Guided Development of Covalent and Mutant-Selective Pyrazolopyrimidines to Target T790M Drug Resistance in Epidermal Growth Factor Receptor.
J. Med. Chem., 60 (18).
S. 7725 - 7745.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
Fang, Zhizhou, Simard, Jeffrey R., Plenker, Dennis, Nguyen, Hoang D., Wolle, Patrik, Baumeister, Stefan and Rauh, Daniel ORCID: 0000-0002-1970-7642
(2015).
Discovery of Inter-Domain Stabilizers-A Novel Assay System for Allosteric Akt Inhibitors.
ACS Chem. Biol., 10 (1).
S. 279 - 289.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1554-8937
Fassunke, Jana, Mueller, Fabienne, Keul, Marina, Michels, Sebastian, Dammert, Marcel A., Schmitt, Anna, Plenker, Dennis, Lategahn, Jonas ORCID: 0000-0001-5993-7082, Heydt, Carina, Braegelmann, Johannes, Tumbrink, Hannah L., Alber, Yannic, Klein, Sebastian, Heimsoeth, Alena, Dahmen, Ilona, Fischers, Rieke N., Scheffler, Matthias, Ihle, Michaela A., Priesner, Vanessa, Scheel, Andreas H., Wagener, Svenja, Kron, Anna, Frank, Konrad, Garbert, Katia, Persigehl, Thorsten, Puesken, Michael, Haneder, Stefan, Schaaf, Bernhard, Rodermann, Ernst, Engel-Riedel, Walburga, Felip, Enriqueta, Smit, Egbert F., Merkelbach-Bruse, Sabine, Reinhardt, H. Christian, Kast, Stefan M., Wolf, Juergen, Rauh, Daniel, Buettner, Reinhard and Sos, Martin L.
(2018).
Overcoming EGFR(G724S)-mediated osimertinib resistance through unique binding characteristics of second-generation EGFR inhibitors.
Nat. Commun., 9.
LONDON:
NATURE PUBLISHING GROUP.
ISSN 2041-1723
Halekotte, Jakob, Witt, Lydia, Ianes, Chiara, Krueger, Marc, Buehrmann, Mike, Rauh, Daniel, Pichlo, Christian, Brunstein, Elena, Luxenburger, Andreas ORCID: 0000-0002-7574-8027, Baumann, Ulrich, Knippschild, Uwe, Bischof, Joachim and Peifer, Christian
(2017).
Optimized 4,5-Diarylimidazoles as Potent/Selective Inhibitors of Protein Kinase CK1 delta and Their Structural Relation to p38 alpha MAPK.
Molecules, 22 (4).
BASEL:
MDPI AG.
ISSN 1420-3049
Heuckmann, Johannes M., Hoelzel, Michael, Sos, Martin L., Heynck, Stefanie, Balke-Want, Hyatt, Koker, Mirjam, Peifer, Martin ORCID: 0000-0002-5243-5503, Weiss, Jonathan, Lovly, Christine M., Gruetter, Christian, Rauh, Daniel
ORCID: 0000-0002-1970-7642, Pao, William and Thomas, Roman K.
(2011).
ALK Mutations Conferring Differential Resistance to Structurally Diverse ALK Inhibitors.
Clin. Cancer Res., 17 (23).
S. 7394 - 7402.
PHILADELPHIA:
AMER ASSOC CANCER RESEARCH.
ISSN 1078-0432
Heuckmann, Johannes M., Rauh, Daniel ORCID: 0000-0002-1970-7642 and Thomas, Roman K.
(2012).
Epidermal Growth Factor Receptor (EGFR) Signaling and Covalent EGFR Inhibition in Lung Cancer.
J. Clin. Oncol., 30 (27).
S. 3417 - 3421.
ALEXANDRIA:
AMER SOC CLINICAL ONCOLOGY.
ISSN 0732-183X
Lategahn, Jonas ORCID: 0000-0001-5993-7082, Keul, Marina, Kloevekorn, Philip, Tumbrink, Hannah L., Niggenaber, Janina
ORCID: 0000-0003-2942-263X, Mueller, Matthias P., Hodson, Luke, Flasshoff, Maren, Hardick, Julia, Grabe, Tobias, Engel, Julian, Schultz-Fademrecht, Carsten, Baumann, Matthias, Ketzer, Julia, Muehlenberg, Thomas, Hiller, Wolf, Guenther, Georgia, Unger, Anke, Mueller, Heiko, Heimsoeth, Alena, Golz, Christopher, Blank-Landeshammer, Bernhard, Kollipara, Laxmikanth, Zahedi, Rene P., Strohmann, Carsten
ORCID: 0000-0002-4787-2135, Hengstler, Jan G., van Otterlo, Willem A. L., Bauer, Sebastian
ORCID: 0000-0001-5949-8120 and Rauh, Daniel
(2019).
Inhibition of osimertinib-resistant epidermal growth factor receptor EGFR-T790M/C797S.
Chem. Sci., 10 (46).
S. 10789 - 10802.
CAMBRIDGE:
ROYAL SOC CHEMISTRY.
ISSN 2041-6539
Lategahn, Jonas, Tumbrink, Hannah L., Schultz-Fademrecht, Carsten, Heimsoeth, Alena, Werr, Lisa ORCID: 0000-0002-3697-4136, Niggenaber, Janina, Keul, Marina, Parmaksiz, Fatma
ORCID: 0009-0003-3771-7128, Baumann, Matthias, Menninger, Sascha, Zent, Eldar, Landel, Ina, Weisner, Joern, Jeyakumar, Kirujan
ORCID: 0000-0002-0184-6775, Heyden, Leonie, Russ, Nicole, Mueller, Fabienne, Lorenz, Carina, Braegelmann, Johannes, Spille, Inga, Grabe, Tobias
ORCID: 0000-0002-8287-1971, Mueller, Matthias P., Heuckmann, Johannes M., Klebl, Bert M., Nussbaumer, Peter, Sos, Martin L. and Rauh, Daniel
(2022).
Insight into Targeting Exon20 Insertion Mutations of the Epidermal Growth Factor Receptor with Wild Type-Sparing Inhibitors.
J. Med. Chem., 65 (9).
S. 6643 - 6656.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1520-4804
Malchers, Florian, Dietlein, Felix, Schottle, Jakob, Lu, Xin, Nogova, Lucia, Albus, Kerstin, Fernandez-Cuesta, Lynnette ORCID: 0000-0002-0724-6703, Heuckmann, Johannes M., Gautschi, Oliver, Diebold, Joachim, Plenker, Dennis, Gardizi, Masyar, Er, Matthias Scheffl, Bos, Marc, Seidel, Danila, Leenders, Frauke, Richters, Andre, Peifer, Martin
ORCID: 0000-0002-5243-5503, Florin, Alexandra, Mainkar, Prathama S., Karre, Nagaraju, Chandrasekhar, Srivari, George, Julie, Silling, Steffi, Rauh, Daniel
ORCID: 0000-0002-1970-7642, Zander, Thomas, Ullrich, Roland T., Reinhardt, H. Christian, Ringeisen, Francois, Buettner, Reinhard, Heukamp, Lukas C., Wolf, Juergen and Thomas, Roman K.
(2014).
Cell-Autonomous and Non-Cell-Autonomous Mechanisms of Transformation by Amplified FGFR1 in Lung Cancer.
Cancer Discov., 4 (2).
S. 246 - 258.
PHILADELPHIA:
AMER ASSOC CANCER RESEARCH.
ISSN 2159-8290
Peifer, Martin ORCID: 0000-0002-5243-5503, Fernandez-Cuesta, Lynnette
ORCID: 0000-0002-0724-6703, Sos, Martin L., George, Julie, Seidel, Danila
ORCID: 0000-0003-4388-3117, Kasper, Lawryn H., Plenker, Dennis, Leenders, Frauke, Sun, Ruping, Zander, Thomas, Menon, Roopika, Koker, Mirjam, Dahmen, Ilona, Mueller, Christian, Di Cerbo, Vincenzo
ORCID: 0000-0002-2920-1274, Schildhaus, Hans-Ulrich, Altmueller, Janine, Baessmann, Ingelore, Becker, Christian, de Wilde, Bram, Vandesompele, Jo
ORCID: 0000-0001-6274-0184, Boehm, Diana, Ansen, Sascha, Gabler, Franziska, Wilkening, Ines, Heynck, Stefanie, Heuckmann, Johannes M., Lu, Xin, Carter, Scott L., Cibulskis, Kristian, Banerji, Shantanu, Getz, Gad, Park, Kwon-Sik, Rauh, Daniel
ORCID: 0000-0002-1970-7642, Gruetter, Christian, Fischer, Matthias, Pasqualucci, Laura, Wright, Gavin
ORCID: 0000-0002-7000-9305, Wainer, Zoe, Russell, Prudence, Petersen, Iver, Chen, Yuan, Stoelben, Erich, Ludwig, Corinna, Schnabel, Philipp, Hoffmann, Hans, Muley, Thomas, Brockmann, Michael, Engel-Riedel, Walburga, Muscarella, Lucia A., Fazio, Vito M., Groen, Harry, Timens, Wim
ORCID: 0000-0002-4146-6363, Sietsma, Hannie, Thunnissen, Erik
ORCID: 0000-0001-5355-8508, Smit, Egbert, Heideman, Danielle A. M., Snijders, Peter J. F., Cappuzzo, Federico, Ligorio, Claudia, Damiani, Stefania, Field, John, Solberg, Steinar, Brustugun, Odd Terje, Lund-Iversen, Marius, Saenger, Joerg, Clement, Joachim H.
ORCID: 0000-0002-6601-2456, Soltermann, Alex, Moch, Holger, Weder, Walter, Solomon, Benjamin, Soria, Jean-Charles, Validire, Pierre, Besse, Benjamin
ORCID: 0000-0001-5090-8189, Brambilla, Elisabeth, Brambilla, Christian, Lantuejoul, Sylvie, Lorimier, Philippe, Schneider, Peter M.
ORCID: 0000-0003-0744-2349, Hallek, Michael, Pao, William, Meyerson, Matthew
ORCID: 0000-0002-9133-8108, Sage, Julien, Shendure, Jay
ORCID: 0000-0002-1516-1865, Schneider, Robert, Buettner, Reinhard, Wolf, Juergen, Nuernberg, Peter, Perner, Sven, Heukamp, Lukas C., Brindle, Paul K., Haas, Stefan
ORCID: 0000-0003-3418-3688 and Thomas, Roman K.
(2012).
Integrative genome analyses identify key somatic driver mutations of small-cell lung cancer.
Nature Genet., 44 (10).
S. 1104 - 1113.
NEW YORK:
NATURE PUBLISHING GROUP.
ISSN 1546-1718
Richters, Andre, Basu, Debjit, Engel, Julian, Ercanoglu, Meryem S., Balke-Want, Hyatt, Tesch, Roberta, Thomas, Roman K. and Rauh, Daniel ORCID: 0000-0002-1970-7642
(2015).
Identification and Further Development of Potent TBK1 Inhibitors.
ACS Chem. Biol., 10 (1).
S. 289 - 299.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1554-8937
Schehr, Miriam, Ianes, Chiara, Weisner, Joern, Heintze, Linda, Mueller, Matthias P., Pichlo, Christian, Charl, Julia, Brunstein, Elena, Ewert, Julia, Lehr, Marc, Baumann, Ulrich, Rauh, Daniel, Knippschild, Uwe, Peifer, Christian and Herges, Rainer (2019). 2-Azo-, 2-diazocine-thiazols and 2-azo-imidazoles as photoswitchable kinase inhibitors: limitations and pitfalls of the photoswitchable inhibitor approach. Photochem. Photobiol. Sci., 18 (6). S. 1398 - 1408. CAMBRIDGE: ROYAL SOC CHEMISTRY. ISSN 1474-9092
Schoettle, Jakob, Chatterjee, Sampurna, Volz, Caroline, Siobal, Maike, Florin, Alexandra, Rokitta, Dennis, Hinze, Yvonne, Dietlein, Felix, Plenker, Dennis, Koenig, Katharina, Albus, Kerstin, Heuckmann, Johannes M., Rauh, Daniel ORCID: 0000-0002-1970-7642, Franz, Thomas, Neumaier, Bernd
ORCID: 0000-0001-5425-3116, Fuhr, Uwe, Heukamp, Lukas C. and Ullrich, Roland T.
(2015).
Intermittent high-dose treatment with erlotinib enhances therapeutic efficacy in EGFR-mutant lung cancer.
Oncotarget, 6 (36).
S. 38458 - 38469.
ORCHARD PARK:
IMPACT JOURNALS LLC.
ISSN 1949-2553
Sos, Martin L., Dietlein, Felix, Peifer, Martin ORCID: 0000-0002-5243-5503, Schoettle, Jakob, Balke-Want, Hyatt, Mueller, Christian, Koker, Mirjam, Richters, Andre, Heynck, Stefanie, Malchers, Florian, Heuckmann, Johannes M., Seidel, Danila, Eyers, Patrick A., Ullrich, Roland T., Antonchick, Andrey P., Vintonyak, Viktor V., Schneider, Peter M.
ORCID: 0000-0003-0744-2349, Ninomiya, Takashi, Waldmann, Herbert
ORCID: 0000-0002-9606-7247, Buettner, Reinhard, Rauh, Daniel
ORCID: 0000-0002-1970-7642, Heukamp, Lukas C. and Thomas, Roman K.
(2012).
A framework for identification of actionable cancer genome dependencies in small cell lung cancer.
Proc. Natl. Acad. Sci. U. S. A., 109 (42).
S. 17034 - 17040.
WASHINGTON:
NATL ACAD SCIENCES.
ISSN 0027-8424
Tueckmantel, Sandra, Greul, Joerg N., Janning, Petra, Brockmeyer, Andreas, Gruetter, Christian, Simard, Jeffrey R., Gutbrod, Oliver, Beck, Michael E., Tietjen, Klaus, Rauh, Daniel ORCID: 0000-0002-1970-7642 and Schreier, Peter H.
(2011).
Identification of Ustilago maydis Aurora Kinase As a Novel Antifungal Target.
ACS Chem. Biol., 6 (9).
S. 926 - 934.
WASHINGTON:
AMER CHEMICAL SOC.
ISSN 1554-8937
Volz, Caroline, Breid, Sara, Selenz, Carolin, Zaplatina, Alina, Golfmann, Kristina, Meder, Lydia, Dietlein, Felix, Borchmann, Sven, Chatterjee, Sampurna, Siobal, Maike, Schoettle, Jakob, Florin, Alexandra, Koker, Mirjam, Nill, Marieke, Ozretic, Luka, Uhlenbrock, Niklas, Smith, Steven, Buettner, Reinhard, Miao, Hui, Wang, Bingcheng, Reinhardt, H. Christian, Rauh, Daniel, Hallek, Michael, Acker-Palmer, Amparo, Heukamp, Lukas C. and Ullrich, Roland T. (2020). Inhibition of Tumor VEGFR2 Induces Serine 897 EphA2-Dependent Tumor Cell Invasion and Metastasis in NSCLC. Cell Reports, 31 (4). CAMBRIDGE: CELL PRESS. ISSN 2211-1247
Weiss, Jonathan, Sos, Martin L., Seidel, Danila, Peifer, Martin ORCID: 0000-0002-5243-5503, Zander, Thomas, Heuckmann, Johannes M., Ullrich, Roland T., Menon, Roopika, Maier, Sebastian, Soltermann, Alex, Moch, Holger, Wagener, Patrick, Fischer, Florian, Heynck, Stefanie, Koker, Mirjam, Schoettle, Jakob, Leenders, Frauke, Gabler, Franziska, Dabow, Ines, Querings, Silvia, Heukamp, Lukas C., Balke-Want, Hyatt, Ansen, Sascha, Rauh, Daniel
ORCID: 0000-0002-1970-7642, Baessmann, Ingelore, Altmueller, Janine, Wainer, Zoe, Conron, Matthew, Wright, Gavin
ORCID: 0000-0002-7000-9305, Russell, Prudence, Solomon, Ben, Brambilla, Elisabeth, Brambilla, Christian, Lorimier, Philippe, Sollberg, Steinar, Brustugun, Odd Terje, Engel-Riedel, Walburga, Ludwig, Corinna, Petersen, Iver, Saenger, Joerg, Clement, Joachim, Groen, Harry, Timens, Wim
ORCID: 0000-0002-4146-6363, Sietsma, Hannie, Thunnissen, Erik
ORCID: 0000-0001-5355-8508, Smit, Egbert, Heideman, Danielle, Cappuzzo, Federico, Ligorio, Claudia, Damiani, Stefania, Hallek, Michael, Beroukhim, Rameen, Pao, William, Klebl, Bert, Baumann, Matthias, Buettner, Reinhard, Ernestus, Karen, Stoelben, Erich, Wolf, Juergen, Nuernberg, Peter, Perner, Sven and Thomas, Roman K.
(2010).
Frequent and Focal FGFR1 Amplification Associates with Therapeutically Tractable FGFR1 Dependency in Squamous Cell Lung Cancer.
Sci. Transl. Med., 2 (62).
WASHINGTON:
AMER ASSOC ADVANCEMENT SCIENCE.
ISSN 1946-6242