Universität zu Köln

2023

Hoffmann, Chris, Kolks, Niklas ORCID: 0000-0001-8532-0684, Smets, Daniel, Haseloer, Alexander ORCID: 0000-0003-0480-7568, Groener, Benedikt, Urusova, Elizaveta A., Endepols, Heike, Neumaier, Felix, Ruschewitz, Uwe ORCID: 0000-0002-6511-6894, Klein, Axel ORCID: 0000-0003-0093-9619, Neumaier, Bernd and Zlatopolskiy, Boris D. (2023). Next Generation Copper Mediators for the Efficient Production of F-18-Labeled Aromatics. Chem.-Eur. J., 29 (2). WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1521-3765

2022

Endepols, Heike, Anglada-Huguet, Marta, Mandelkow, Eckhard, Schmidt, Yannick, Krapf, Philipp, Zlatopolskiy, Boris D., Neumaier, Bernd ORCID: 0000-0001-5425-3116, Mandelkow, Eva-Maria and Drzezga, Alexander (2022). Assessment of the In Vivo Relationship Between Cerebral Hypometabolism, Tau Deposition, TSPO Expression, and Synaptic Density in a Tauopathy Mouse Model: a Multi-tracer PET Study. Mol. Neurobiol., 59 (6). S. 3402 - 3414. NEW YORK: SPRINGER. ISSN 1559-1182

Endepols, Heike, Zlatopolskiy, Boris D., Zischler, Johannes, Alavinejad, Nazanin, Apetz, Nadine ORCID: 0000-0003-3232-2517, Vus, Stefanie, Drzezga, Alexander and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2022). Imaging of cerebral tryptophan metabolism using 7-[F-18]FTrp-PET in a unilateral Parkinsonian rat model. Neuroimage, 247. SAN DIEGO: ACADEMIC PRESS INC ELSEVIER SCIENCE. ISSN 1095-9572

Walter, Nils ORCID: 0000-0003-3727-3750, Bertram, Jan, Drewes, Birte ORCID: 0000-0002-6849-1438, Bahutski, Victor, Timmer, Marco, Schuetz, Markus B., Kraemer, Felicia, Neumaier, Felix, Endepols, Heike, Neumaier, Bernd and Zlatopolskiy, Boris D. (2022). Convenient PET-tracer production via SuFEx F-18-fluorination of nanomolar precursor amounts. Eur. J. Med. Chem., 237. ISSY-LES-MOULINEAUX: ELSEVIER FRANCE-EDITIONS SCIENTIFIQUES MEDICALES ELSEVIER. ISSN 1768-3254

2021

Hoffmann, Chris ORCID: 0000-0003-1093-0183, Evcueman, Sibel, Neumaier, Felix ORCID: 0000-0002-6376-6391, Zlatopolskiy, Boris D., Humpert, Swen ORCID: 0000-0002-1995-0714, Bier, Dirk, Holschbach, Marcus, Schulze, Annette, Endepols, Heike and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2021). [F-18]ALX5406: A Brain-Penetrating Prodrug for GlyT1-Specific PET Imaging. ACS Chem. Neurosci., 12 (18). S. 3335 - 3347. WASHINGTON: AMER CHEMICAL SOC. ISSN 1948-7193

Humpert, Swen ORCID: 0000-0002-1995-0714, Omrane, Mohamed A., Urusova, Elizaveta A., Gremer, Lothar ORCID: 0000-0001-7065-5027, Willbold, Dieter ORCID: 0000-0002-0065-7366, Endepols, Heike, Krasikova, Raisa N., Neumaier, Bernd ORCID: 0000-0001-5425-3116 and Zlatopolskiy, Boris D. (2021). Rapid F-18-labeling via Pd-catalyzed S-arylation in aqueous medium. Chem. Commun., 57 (29). S. 3547 - 3551. CAMBRIDGE: ROYAL SOC CHEMISTRY. ISSN 1364-548X

Kraemer, Felicia, Groener, Benedikt, Hoffmann, Chris, Craig, Austin, Brugger, Melanie, Drzezga, Alexander, Timmer, Marco, Neumaier, Felix, Zlatopolskiy, Boris D., Endepols, Heike and Neumaier, Bernd (2021). Evaluation of 3-l- and 3-d-[F-18]Fluorophenylalanines as PET Tracers for Tumor Imaging. Cancers, 13 (23). BASEL: MDPI. ISSN 2072-6694

Neumaier, Felix ORCID: 0000-0002-6376-6391, Zlatopolskiy, Boris D. and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2021). Drug Penetration into the Central Nervous System: Pharmacokinetic Concepts and In Vitro Model Systems. Pharmaceutics, 13 (10). BASEL: MDPI. ISSN 1999-4923

Orlovskaya, Viktoriya V., Craig, Austin S., Fedorova, Olga S., Kuznetsova, Olga F., Neumaier, Bernd ORCID: 0000-0001-5425-3116, Krasikova, Raisa N. and Zlatopolskiy, Boris D. (2021). Production of 6-l-[F-18]Fluoro-m-tyrosine in an Automated Synthesis Module for C-11-Labeling. Molecules, 26 (18). BASEL: MDPI. ISSN 1420-3049

Schroeder, Daniel C., Popp, Erik, Rohleder, Cathrin ORCID: 0000-0002-3559-1846, Vus, Stefanie, Bethencourt, David de la Puente, Finke, Simon R., Zlatopolskiy, Boris D., Zischler, Johannes, Drzezga, Alexander ORCID: 0000-0001-6018-716X, Herff, Holger, Annecke, Thorsten, Hucho, Tim ORCID: 0000-0002-4147-9308, Neumaier, Bernd, Boettiger, Bernd W. and Endepols, Heike (2021). Positron Emission Tomography Imaging of Long-Term Expression of the 18 kDa Translocator Protein After Sudden Cardiac Arrest in Rats. Shock, 55 (5). S. 620 - 630. PHILADELPHIA: LIPPINCOTT WILLIAMS & WILKINS. ISSN 1540-0514

2020

Craig, Austin, Kolks, Niklas, Urusova, Elizaveta A., Zischler, Johannes, Brugger, Melanie, Endepols, Heike, Neumaier, Bernd ORCID: 0000-0001-5425-3116 and Zlatopolskiy, Boris D. (2020). Preparation of labeled aromatic amino acidsvialate-stage(18)F-fluorination of chiral nickel and copper complexes. Chem. Commun., 56 (66). S. 9505 - 9509. CAMBRIDGE: ROYAL SOC CHEMISTRY. ISSN 1364-548X

Dietlein, Felix, Hohberg, Melanie, Kobe, Carsten, Zlatopolskiy, Boris D., Krapf, Philipp, Endepols, Heike ORCID: 0000-0002-6166-4818, Taeger, Philipp, Hammes, Jochen, Heidenreich, Axel, Neumaier, Bernd, Drzezga, Alexander and Dietlein, Markus (2020). An F-18-Labeled PSMA Ligand for PET/CT of Prostate Cancer: First-in-Humans Observational Study and Clinical Experience with F-18-JK-PSMA-7 During the First Year of Application. J. Nucl. Med., 61 (2). S. 202 - 210. RESTON: SOC NUCLEAR MEDICINE INC. ISSN 1535-5667

Dietlein, Felix, Kobe, Carsten, Hohberg, Melanie, Zlatopolskiy, Boris D., Krapf, Philipp, Endepols, Heike, Taeger, Philipp, Hammes, Jochen ORCID: 0000-0003-2850-9450, Heidenreich, Axel, Persigehl, Thorsten, Neumaier, Bernd, Drzezga, Alexander and Dietlein, Markus (2020). Intraindividual Comparison of F-18-PSMA-1007 with Renally Excreted PSMA Ligands for PSMA PET Imaging in Patients with Relapsed Prostate Cancer. J. Nucl. Med., 61 (5). S. 729 - 735. RESTON: SOC NUCLEAR MEDICINE INC. ISSN 1535-5667

Neumaier, Felix ORCID: 0000-0002-6376-6391, Zlatopolskiy, Boris D. and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2020). Nuclear Medicine in Times of COVID-19: How Radiopharmaceuticals Could Help to Fight the Current and Future Pandemics. Pharmaceutics, 12 (12). BASEL: MDPI. ISSN 1999-4923

Zlatopolskiy, Boris D., Endepols, Heike, Krasikova, Raisa N., Fedorova, Olga S., Ermert, Johannes ORCID: 0000-0002-2561-7766 and Neumaier, Bernd (2020). C-11- and F-18-labelled tryptophans as PET-tracers for imaging of altered tryptophan metabolism in age-associated disorders. Russ. Chem. Rev., 89 (9). S. 879 - 897. BRISTOL: TURPION LTD. ISSN 1468-4837

Zlatopolskiy, Boris D., Neumaier, Felix ORCID: 0000-0002-6376-6391, Ruengeler, Till, Drewes, Birte ORCID: 0000-0002-6849-1438, Kolks, Niklas ORCID: 0000-0001-8532-0684 and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2020). Preparation of a First(18)F-Labeled Agonist for M(1)Muscarinic Acetylcholine Receptors. Molecules, 25 (12). BASEL: MDPI. ISSN 1420-3049

2019

Endepols, Heike ORCID: 0000-0002-6166-4818, Morgenroth, Agnieszka, Zlatopolskiy, Boris D., Krapf, Philipp ORCID: 0000-0003-1671-2443, Zischler, Johannes, Richarz, Raphael, Vasquez, Sergio Munoz, Neumaier, Bernd ORCID: 0000-0001-5425-3116 and Mottaghy, Felix M. (2019). Peripheral ganglia in healthy rats as target structures for the evaluation of PSMA imaging agents. BMC Cancer, 19. LONDON: BMC. ISSN 1471-2407

Hohberg, Melanie, Kobe, Carsten, Krapf, Philipp ORCID: 0000-0003-1671-2443, Taeger, Philipp, Hammes, Jochen, Dietlein, Felix, Zlatopolskiy, Boris D., Endepolst, Heike, Wild, Markus, Neubauer, Stephan, Heidenreich, Axel, Neumaier, Bernd, Drzezga, Alexander and Dietlein, Markus (2019). Biodistribution and radiation dosimetry of [F-18]-JK-PSMA-7 as a novel prostate-specific membrane antigen-specific ligand for PET/CT imaging of prostate cancer. EJNMMI Res., 9. LONDON: SPRINGEROPEN. ISSN 2191-219X

Modemann, Daniel J., Zlatopolskiy, Boris D., Urusova, Elizaveta A., Zischler, Johannes, Craig, Austin, Ermert, Johannes ORCID: 0000-0002-2561-7766, Guliyev, Mehrab, Endepols, Heike ORCID: 0000-0002-6166-4818 and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2019). 2-[F-18] Fluorophenylalanine: Synthesis by Nucleophilic F-18-Fluorination and Preliminary Biological Evaluation. Synthesis, 51 (3). S. 664 - 677. STUTTGART: GEORG THIEME VERLAG KG. ISSN 1437-210X

Orlovskaya, Victoriya V., Modemann, Daniel J., Kuznetsova, Olga F., Fedorova, Olga S. ORCID: 0000-0002-9122-9622, Urusova, Elizaveta A., Kolks, Niklas ORCID: 0000-0001-8532-0684, Neumaier, Bernd ORCID: 0000-0001-5425-3116, Krasikova, Raisa N. and Zlatopolskiy, Boris D. (2019). Alcohol-Supported Cu-Mediated F-18-Fluorination of Iodonium Salts under Minimalist Conditions. Molecules, 24 (17). BASEL: MDPI. ISSN 1420-3049

Zlatopolskiy, Boris D., Endepols, Heike ORCID: 0000-0002-6166-4818, Krapf, Philipp ORCID: 0000-0003-1671-2443, Guliyev, Mehrab, Urusova, Elizaveta A., Richarz, Raphael, Hohberg, Melanie, Dietlein, Markus, Drzezga, Alexander and Neumaier, Bernd (2019). Discovery of F-18-JK-PSMA-7, a PET Probe for the Detection of Small PSMA-Positive Lesions. J. Nucl. Med., 60 (6). S. 817 - 824. RESTON: SOC NUCLEAR MEDICINE INC. ISSN 1535-5667

Zlatopolskiy, Boris D., Zischler, Johannes ORCID: 0000-0003-3996-7473, Krapf, Philipp ORCID: 0000-0003-1671-2443, Richarz, Raphael, Lauchner, Katharina and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2019). Minimalist approach meets green chemistry: Synthesis of F-18- labeled (hetero)aromatics in pure ethanol. J. Label. Compd. Radiopharm., 62 (8). S. 404 - 411. HOBOKEN: WILEY. ISSN 1099-1344

2018

Endepols, Heike ORCID: 0000-0002-6166-4818, Mottaghy, Felix M., Simsekyilmaz, Sakine, Bucerius, Jan, Vogt, Felix, Winz, Oliver, Richarz, Raphael, Krapf, Philipp ORCID: 0000-0003-1671-2443, Neumaier, Bernd ORCID: 0000-0001-5425-3116, Zlatopolskiy, Boris D. and Morgenroth, Agnieszka (2018). In vivo Molecular Imaging of Glutamate Carboxypeptidase II Expression in Re-endothelialisation after Percutaneous Balloon Denudation in a Rat Model. Sci Rep, 8. LONDON: NATURE PUBLISHING GROUP. ISSN 2045-2322

2017

Dietlein, Felix, Kobe, Carsten, Neubauer, Stephan, Schmidt, Matthias, Stockter, Simone, Fischer, Thomas, Schomaecker, Klaus, Heidenreich, Axel, Zlatopolskiy, Boris D., Neumaier, Bernd ORCID: 0000-0001-5425-3116, Drzezga, Alexander and Dietlein, Markus (2017). PSA-Stratified Performance of F-18- and Ga-68-PSMA PET in Patients with Biochemical Recurrence of Prostate Cancer. J. Nucl. Med., 58 (6). S. 947 - 953. RESTON: SOC NUCLEAR MEDICINE INC. ISSN 1535-5667

Feni, Lucia, Omrane, M. Aymen, Fischer, Moritz, Zlatopolskiy, Boris D., Neumaier, Bernd ORCID: 0000-0001-5425-3116 and Neundorf, Ines ORCID: 0000-0001-6450-3991 (2017). Convenient Preparation of F-18-Labeled Peptide Probes for Potential Claudin-4 PET Imaging. Pharmaceuticals, 10 (4). BASEL: MDPI. ISSN 1424-8247

Morgenroth, Agnieszka, Vogg, Andreas T. J., Neumaier, Bernd ORCID: 0000-0001-5425-3116, Mottaghy, Felix M. and Zlatopolskiy, Boris D. (2017). Radioiodinated indomethacin amide for molecular imaging of cyclooxygenase-2 expressing tumors. Oncotarget, 8 (11). S. 18059 - 18070. ORCHARD PARK: IMPACT JOURNALS LLC. ISSN 1949-2553

Zarrad, Fadi, Zlatopolskiy, Boris D., Krapf, Philipp ORCID: 0000-0003-1671-2443, Zischler, Johannes ORCID: 0000-0003-3996-7473 and Neumaier, Bernd (2017). A Practical Method for the Preparation of 18F-Labeled Aromatic Amino Acids from Nucleophilic [18F]Fluoride and Stannyl Precursors for Electrophilic Radiohalogenation. Molecules, 22 (12). BASEL: MDPI. ISSN 1420-3049

Zischler, Johannes ORCID: 0000-0003-3996-7473, Kolks, Niklas, Modemann, Daniel, Neumaier, Bernd ORCID: 0000-0001-5425-3116 and Zlatopolskiy, Boris D. (2017). Alcohol-Enhanced Cu-Mediated Radiofluorination. Chem.-Eur. J., 23 (14). S. 3251 - 3257. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1521-3765

2016

Krapf, Philipp ORCID: 0000-0003-1671-2443, Richarz, Raphael, Urusova, Elizaveta A., Neumaier, Bernd ORCID: 0000-0001-5425-3116 and Zlatopolskiy, Boris D. (2016). Seyferth-Gilbert Homologation as a Route to F-18-Labeled Building Blocks: Preparation of Radiofluorinated Phenylacetylenes and Their Application in PET Chemistry. Eur. J. Org. Chem., 2016 (3). S. 430 - 434. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1099-0690

Zischler, Johannes ORCID: 0000-0003-3996-7473, Krapf, Philipp ORCID: 0000-0003-1671-2443, Richarz, Raphael, Zlatopolskiy, Boris D. and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2016). Automated synthesis of 4-[F-18]fluoroanisole, [F-18]DAA1106 and 4-[F-18]FPhe using Cu-mediated radiofluorination under minimalist conditions. Appl. Radiat. Isot., 115. S. 133 - 138. OXFORD: PERGAMON-ELSEVIER SCIENCE LTD. ISSN 0969-8043

2015

Dietlein, Markus, Kobe, Carsten, Kuhnert, Georg, Stockter, Simone, Fischer, Thomas, Schomaecker, Klaus, Schmidt, Matthias, Dietlein, Felix, Zlatopolskiy, Boris D., Krapf, Philipp, Richarz, Raphael, Neubauer, Stephan, Drzezga, Alexander and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2015). Comparison of [F-18]DCFPyL and [Ga-68]Ga-PSMA-HBED-CC for PSMA-PET Imaging in Patients with Relapsed Prostate Cancer. Mol. Imaging. Biol., 17 (4). S. 575 - 585. NEW YORK: SPRINGER. ISSN 1860-2002

Zlatopolskiy, Boris D., Zischler, Johannes ORCID: 0000-0003-3996-7473, Urusova, Elizaveta A., Endepols, Heike ORCID: 0000-0002-6166-4818, Kordys, Elena, Frauendorf, Holm, Mottaghy, Felix M. and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2015). A Practical One-Pot Synthesis of Positron Emission Tomography (PET) Tracers via Nickel-Mediated Radiofluorination. ChemistryOpen, 4 (4). S. 457 - 463. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 2191-1363

2014

Morgenroth, Agnieszka, Vogg, Andreas T. J., Zlatopolskiy, Boris D., Siluschek, Monika, Oedekoven, Caroline and Mottaghy, Felix M. (2014). Breaking the Invulnerability of Cancer Stem Cells: Two-Step Strategy to Kill the Stem-like Cell Subpopulation of Multiple Myeloma. Mol. Cancer Ther., 13 (1). S. 144 - 154. PHILADELPHIA: AMER ASSOC CANCER RESEARCH. ISSN 1538-8514

Zlatopolskiy, Boris D., Krapf, Philipp, Richarz, Raphael, Frauendorf, Holm, Mottaghy, Felix M. and Neumaier, Bernd ORCID: 0000-0001-5425-3116 (2014). Synthesis of F-18-Labelled beta-Lactams by Using the Kinugasa Reaction. Chem.-Eur. J., 20 (16). S. 4697 - 4704. WEINHEIM: WILEY-V C H VERLAG GMBH. ISSN 1521-3765